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CP-96345CP-96345是具有抗炎作用的P物质拮抗剂,由辉瑞公司研究。本品可用于治疗神经性炎症。它的对映体CP-96344体外试验不具有NK1受体拮抗剂的活性,但对血流动力学和心血管组织收缩的作用类似,这表明CP-96345的心血管作用可能与...
CP-96345CP-96345 is an anti-inflammatory substance P antagonist studied by Pfizer. This product can be used to treat neurological inflammation. Its enantiomer CP-96344 in vitro test does not have the activity of an NK1 receptor antagonist, but has similar effects on hemodynamics and cardiovascular tissue contractility, suggesting that the cardiovascular effects of CP-96345 may be related to ...