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N-(6-(2-甲氧基-3-(4-氟苯磺酰氨基)-5-吡啶基-2-[1,2,4]三唑[1,5-a]吡啶基乙酰胺(A)具有优异的抗肿瘤活性[1],但是其毒性较大。
1-烷基-3-(6-(2-甲氧基3-磺酰氨基-5-吡啶基-2-[1,2,4]三唑[1,5a]吡啶基)脲类的活性研究
【摘 要】
：
N-(6-(2-甲氧基-3-(4-氟苯磺酰氨基)-5-吡啶基-2-[1,2,4]三唑[1,5-a]吡啶基乙酰胺(A)具有优异的抗肿瘤活性[1],但是其毒性较大。
【机 构】
：
西安交通大学药学院,西安 710061
【出 处】
：
2015年全国药物化学学术会议暨第五届中英药物化学学术会议
【发表日期】
：
2015年3期
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化合物N-(2-氯-5-(2-乙酰氨基-6-苯并噻唑基)-3-吡啶基)-4-氟苯磺酰胺(A)具有优异的抗肿瘤活性[1]，但是其毒性较大。
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